Macitentan

• Description:

  Endothelin (ET)(A) and ET(B) receptor antagonist

• Product Name Alternative:

  5-(4-bromophenyl)-6-[2-(5-bromopyrimidin-2-yl)oxyethoxy]-N-(propylsulfamoyl)pyrimidin-4-amine

• Field of Research:

  GPCR G protein Endothelin Receptor

• Purity:

  0.9953

• Form:

  A solid

• Solubility:

  ≥24.4 mg/mL in DMSO; insoluble in H2O; insoluble in EtOH

• Smiles:

  CCCNS(=O)(=O)NC1=C(C(=NC=N1)OCCOC2=NC=C(C=N2)Br)C3=CC=C(C=C3)Br

• Molecular Formula:

  C19H20Br2N6O4S

• Molecular Weight:

  588.27

• Shipping Conditions:

  Blue ice

• Storage Conditions:

  Store at -20°C.

• CAS Number:

  441798-33-0