BMS-754807

CAT: 0607-A1185-100Size: 100 mgDry Ice: NoHazardous: No

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CAT#:0607-A1185-100Size:100 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Description

IGF-1R/InsR inhibitor,potent and selective

CAS Number

1001350-96-4

Product Name Alternative

(2S)-1-[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl]-N-(6-fluoropyridin-3-yl)-2-methylpyrrolidine-2-carboxamide

Field of Research

Tyrosine Kinase IGF1R

Purity

0.9953

Form

A solid

Solubility

≥23.05 mg/mL in DMSO; insoluble in H2O; ≥27.75 mg/mL in EtOH

Smiles

CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F

Molecular Formula

C23H24FN9O

Molecular Weight

461.49

Shipping Conditions

Blue ice

Storage Conditions

Store at -20°C.

1001350-96-4

PubChem

cas	1001350-96-4
modify	2026-05-17
description	BMS-754807 is a pyrrolotriazine that is pyrrolo[2,1-f][1,2,4]triazine which is substituted at position 2 by the pyrrolidine nitrogen of (2S)-N-(6-fluoropyridin-3-yl)-2-methylprolinamide, and at position 4 by a (5-cyclopropyl-1H-pyrazol-3-yl)amino group. It is a potent, reversible inhibitor of the insulin-like growth factor 1 receptor/insulin receptor family kinases. It has a role as an antineoplastic agent and an EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor. It is a member of pyrazoles, a member of pyridines, a member of pyrrolidines and a pyrrolotriazine.
synonyms	BMS-7548071001350-96-4BMS 754807BMS754807W9E3353E8JBMS-754807-01 (2S)-1-[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl]-N-(6-fluoropyridin-3-yl)-2-methylpyrrolidine-2-carboxamide CHEBI:88339 (2S)-1-{4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}-N-(6-fluoropyridin-3-yl)-2-methylpyrrolidine-2-carboxamide 2-PYRROLIDINECARBOXAMIDE, 1-(4-((5-CYCLOPROPYL-1H-PYRAZOL-3-YL)AMINO)PYRROLO(2,1-F)(1,2,4)TRIAZIN-2-YL)-N-(6-FLUORO-3-PYRIDINYL)-2-METHYL-, (2S)- + 15 more
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Catalog	Name
HY-10200-01	BMS-754807
RM-B131901-01	Bms 754807