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Y06036

CAT: 0804-HY-111502-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-111502-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Y06036 is a potent and selective BET inhibitor, which binds to the BRD4 (1) bromodomain with Kd value of 82 nM[1]. Antitumor activity[1].
CAS Number
1832671-96-1
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Neuroscience-Neuromodulation
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/Y06036.html
Purity
98.57
Solubility
DMSO : 130 mg/mL (ultrasonic)
Smiles
BrC1=CC(S(=O)(NC2=C(OC)C=C(ON=C3C)C3=C2)=O)=C(OC)C=C1
Molecular Formula
C16H15BrN2O5S
Molecular Weight
427.27
Precautions
H302, H315, H319, H335
References & Citations
[1]Zhang M, et al. Structure-Based Discovery and Optimization of Benzo[ d]isoxazole Derivatives as Potent and Selective BET Inhibitors for Potential Treatment of Castration-Resistant Prostate Cancer (CRPC) . J Med Chem. 2018 Apr 12;61 (7) :3037-3058.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
BRD4

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CatalogName
BA4738-100Y06036
A19665-100Y06036 100mg
A19665-5Y06036 5mg
A19665-50Y06036 50mg
A19665-25Y06036 25mg
A19665-10Y06036 10mg
A19665-500Y06036 500mg
A19665-10mM-DY06036 10mM * 1mL in DMSO

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