Tasipimidine

CAT: 0804-HY-109075Size: 1 EachDry Ice: NoHazardous: No

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CAT#:0804-HY-109075Size:1 Each

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Description

Tasipimidine is an orally active and selective α2A-adrenoceptor agonist with a pEC50 of 7.57 for human α2A-adrenoceptors and an EC50 of 5.7 nM for rat α2-adrenoceptor. Tasipimidine can be utilized in research related to situational anxiety and fear[1][2].

CAS Number

1465908-70-6

UNSPSC

12352005

Target

Adrenergic Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/tasipimidine.html

Smiles

COC1=C2CCOC(C3=NCCN3)C2=CC=C1

Molecular Formula

C13H16N2O2

Molecular Weight

232.28

References & Citations

[1]Lehtimäki J, et al. Tasipimidine-the pharmacological profile of a novel orally active selective α2A-adrenoceptor agonist. Eur J Pharmacol. 2022 May 15;923:174949.|[2]Korpivaara M, et al. Tasipimidine, a novel orally administered alpha-2 adrenoceptor agonist, alleviates canine acute anxiety associated with owner departure—A pilot study. Journal of Veterinary Behavior, 2022, 58: 54-61.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

Phase 2

Isoform

α adrenergic receptor

Alternative Products

Catalog	Name
T28924-01	Tasipimidine
T60964-01	Tasipimidine sulfate

Tasipimidine

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