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Ricasetron

CAT: 0804-HY-101709-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-101709-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Ricasetron (BRL-46470) is a selective and orally active 5-HT3 receptor antagonist. Ricasetron displays little or no affinity for a variety of other neurotransmitter receptors. Ricasetron has anxiolytic and antiemetic effects[1][2].
CAS Number
117086-68-7
Product Name Alternative
BRL-46470
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ricasetron.html
Purity
98.62
Solubility
DMSO : 50 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
O=C(N1C(C=CC=C2)=C2C(C)(C)C1)N[C@H]3C[C@@H](CC4)N(C)[C@@H]4C3
Molecular Formula
C19H27N3O
Molecular Weight
313.44
References & Citations
[1]Steward LJ, et al. Evidence that the atypical 5-HT3 receptor ligand, [3H]-BRL46470, labels additional 5-HT3 binding sites compared to [3H]-granisetron. Br J Pharmacol. 1995 Sep;116 (2) :1781-8.|[2]Gao B, et al. Effects of sub-chronic treatment with chlordiazepoxide, buspirone and the 5-HT3 receptor antagonist, BRL 46470, on the social behaviour of mice. Neuropharmacology. 1992 Mar;31 (3) :207-13.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 2
Isoform
5-HT3 Receptor

Alternative Products

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M34396-01Ricasetron
A15499-50Ricasetron 50mg
A15499-10Ricasetron 10mg
A15499-100Ricasetron 100mg
A15499-25Ricasetron 25mg
A15499-5Ricasetron 5mg
A15499-2Ricasetron 2mg
A15499-1Ricasetron 1mg

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