Niraparib metabolite M1
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


Niraparib metabolite M1
UNSPSC Description:
Niraparib metabolite M1 is a metabolite of niraparib, and the latter one acts as a novel poly(ADP-Ribose) polymerase (PARP) inhibitor.Target Antigen:
Drug MetaboliteType:
Reference compoundRelated Pathways:
Metabolic Enzyme/ProteaseField of Research:
OthersAssay Protocol:
https://www.medchemexpress.com/Niraparib-metabolite-M1.htmlPurity:
99.69Solubility:
DMSO : ≥ 100 mg/mLSmiles:
O=C(C1=CC=CC2=CN(C3=CC=C([C@H]4CNCCC4)C=C3)N=C12)OMolecular Weight:
321.37References & Citations:
[1]van Andel L, et al. Liquid chromatography-tandem mass spectrometry assay for the quantification of niraparib and its metabolite M1 in human plasma and urine. J Chromatogr B Analyt Technol Biomed Life Sci. 2016 Nov 19;1040:14-21Shipping Conditions:
Room TemperatureStorage Conditions:
-20°C, 3 years; 4°C, 2 years (Powder)Clinical Information:
No Development ReportedCAS Number:
1476777-06-6
