Tersolisib

CAT: 0804-HY-156681-01Size: 5 mgDry Ice: NoHazardous: No

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CAT#:0804-HY-156681-01Size:5 mg

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Description

STX-478 (compound 80) is an oral CNS-penetrant allosteric mutant-selective PI3Kα inhibitor. STX-478 shows robust and durable tumor regression and can be used in cancer research[1].

CAS Number

2883540-92-7

Product Name Alternative

STX-478

UNSPSC

12352005

Target

PI3K

Type

Reference compound

Related Pathways

PI3K/Akt/mTOR

Applications

Cancer-Kinase/protease

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/stx-478.html

Concentration

10mM

Purity

99.63

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

NC1=NC=C(C=N1)NC(N[C@H](C2=C(C3=CC(F)=CC(F)=C3O2)C)C(F)(F)F)=O

Molecular Formula

C16H12F5N5O2

Molecular Weight

401.29

References & Citations

[1]JR David St Jean, et al. Urea derivatives which can be used to treat cancer. Patent WO2022265993A1.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

Phase 2

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Catalog	Name
C01887-01	Tersolisib (STX-478)

Tersolisib

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