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MZ-1

CAT: 1568-C13753-100mgSize: 100 mgDry Ice: NoHazardous: No
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CAT#:1568-C13753-100mgSize:100 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1797406-69-9
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1=C (SC2=C1C (=NC (C3=NN=C (N32) C) CC (=O) NCCOCCOCCOCC (=O) NC (C (=O) N4CC (CC4C (=O) NCC5=CC=C (C=C5) C6=C (N=CS6) C) O) C (C) (C) C) C7=CC=C (C=C7) Cl) C
Molecular Formula
C49H60ClN9O8S2
Additionnal Information
MZ-1 is a PROTAC degrader of bromodomain-containing protein 4 (BRD4) . MZ-1 binds to the Brd bromodomain with Kd of 62 nM, 60 nM, 21 nM, 13 nM, 39 nM and 15 nM for Brd2BD1, Brd2BD2, Brd3BD1, Brd3BD2, Brd4BD1 and Brd4BD2.
Storage Conditions
3 years -20°C powder