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PLX51107

CAT: 1568-C13630-5mgSize: 5 mgDry Ice: NoHazardous: No
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CAT#:1568-C13630-5mgSize:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1627929-55-8
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1=C (C (=NO1) C) C2=CC3=C (C (=CN3C (C) C4=CC=CC=N4) C5=CC=C (C=C5) C (=O) O) N=C2
Molecular Formula
C26H22N4O3
Additionnal Information
PLX51107 is as a novel BET inhibitor with modest preference for bromodomain-1 (BD1) versus bromodomain-2 (BD2) within each BET protein (Kd = 1.6, 2.1, 1.7, and 5 nM for BD1 and 5.9, 6.2, 6.1 and 120 nM for BD2 of BRD2, BRD3, BRD4, and BRDT, respectively. Among non-BET proteins, PLX51107 shows significant interactions only with the bromodomains of CBP and EP300 (p300) (Kd in the 100 nM range) .
Storage Conditions
3 years -20°C powder

Alternative Products

CatalogName
MBS3842811-01PLX51107
A18345-100PLX51107 100mg
A18345-2PLX51107 2mg
A18345-5PLX51107 5mg
A18345-25PLX51107 25mg
A18345-10PLX51107 10mg
A18345-50PLX51107 50mg
A18345-1PLX51107 1mg
A18345-10mM-DPLX51107 10mM * 1mL in DMSO

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