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EPZ005687

CAT: 1568-C12375-5mgSize: 5 mgDry Ice: YesHazardous: No
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CAT#:1568-C12375-5mgSize:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1396772-26-1
Target
Histone Methyltransferase
Applications
Epigenetics
Smiles
CC1=CC (=C (C (=O) N1) CNC (=O) C2=C3C=NN (C3=CC (=C2) C4=CC=C (C=C4) CN5CCOCC5) C6CCCC6) C
Molecular Formula
C32H37N5O3
Additionnal Information
EPZ005687 is a potent and selective inhibitor of EZH2 with Ki of 24 nM in a cell-free assay, 50-fold selectivity against EZH1 and 500-fold selectivity against 15 other protein methyltransferases.
Storage Conditions
2 years -80 in solvent