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PF 429242

CAT: 1568-C11875-5mgSize: 5 mgDry Ice: NoHazardous: No
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CAT#:1568-C11875-5mgSize:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
947303-87-9
Target
S1P Receptor
Applications
GPCR & G Protein
Smiles
CCN (CC) CC1=CC=C (C=C1) C (=O) N (CCC2=CC=CC=C2OC) C3CCNC3
Molecular Formula
C25H35N3O2
Additionnal Information
PF 429242 is known as a S1P inhibitor with an IC50 of 170 nM, showing no significant inhibition of trypsin, elastase, proteinase K, plasmin, kallikren, factor XIa, thrombin, or furin at concentrations up to 100 μM and only modest inhibition of urokinase (IC50 = 50 μM) and factor Xa (IC50 = 100 μM) .
Storage Conditions
3 years -20°C powder