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Pradigastat

CAT: 1568-C04256-5mgSize: 5 mgDry Ice: NoHazardous: No
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CAT#:1568-C04256-5mgSize:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
956136-95-1
Synonyms
LCQ-908
Target
Acyltransferase
Applications
Metabolism
Molecular Formula
C25H24F3N3O2
Additionnal Information
Pradigastat (LCQ-908) is a potent and selective inhibitor of DGAT1 with an IC50 of 57 nM in hDGAT1. It also inhibits OATP1B1, OATP1B3 , and OAT3 activity in a concentration-dependent manner, with an IC50 of 1.66 μM, 3.34 μM, and 0.973 μM, respectively.