Products for Research Use Only
RegisterLogin

Pitolisant

CAT: 0957-E4955-100mgSize: 100 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0957-E4955-100mgSize:100 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
362665-56-3
Synonyms
BF2.649, Tiprolisant
Target
Histamine Receptor
Applications
Neuronal Signaling
Additionnal Information
Pitolisant (BF2.649, Tiprolisant) is a potent, selective antagonist of the non-imidazole histamine H3 receptor, with a Ki value of 0.16 nM and an EC50 of 1.5 nM as an inverse agonist. It enhances the activity of histaminergic neurons, promoting vigilance and cognitive function. It is useful in research on wakefulness, memory deficits, and cognitive disorders.
Storage Conditions
2 years -20°C liquid

Alternative Products

CatalogName
BA5401-50Pitolisant
A3727-5.1Pitolisant hydrochloride
319900Pitolisant HCl
HY-12199SPitolisant-d10
HY-12199B-01Pitolisant (hydrochloride)
HY-12199APitolisant (oxalate)
T12491-01Pitolisant oxalate

Popular Products