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CP94253

CAT: 0804-HY-103151ASize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-103151ASize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CP94253 is a selective, orally active agonist for serotonin receptor 1B (5-HT1B), through competitive binding with iodocyanopindolol (ICP) to the 5-HT1 receptor. CP94253 binds to the 5-HT1B, 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, with Kis of 2, 89, 49, 860 and 1600 nM. CP94253 causes satiety, anorexia, weight loss and hyperlocomotion in rats model[1].
CAS Number
131084-35-0
UNSPSC
12352005
Hazard Statement
H302-H315-H319-H335
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/cp94253.html
Smiles
CCCOC1=NC2=C(NC=C2C3=CCNCC3)C=C1
Molecular Formula
C15H19N3O
Molecular Weight
257.33
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501
References & Citations
[1]Koe B K, et al., Biochemical and behavioral studies of the 5‐HT1B receptor agonist, CP‐94,253[J]. Drug development research, 1992, 26 (3) : 241-250.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT1 Receptor; mLAG-3; α-1 microglobulin

Alternative Products

CatalogName
T88269-01CP94253
GTR19172637-01CP94253 hydrochloride

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