WH-4-023

CAT: 1568-C17986Size: 100 mgDry Ice: YesHazardous: No
CAT#:1568-C17986Size:100 mg
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
CAS Number
837422-57-8
Synonyms
KIN001-112, KIN112, Dual LCK/SRC inhibitor
SKU
C17986-100mg
Target
Src
Applications
Protein Tyrosine Kinase
Smiles
CC1=C (C (=CC=C1) C) OC (=O) N (C2=C (C=C (C=C2) OC) OC) C3=NC (=NC=C3) NC4=CC=C (C=C4) N5CCN (CC5) C
Molecular Formula
C32H36N6O4
Additionnal Information
WH-4-023 (KIN001-112, KIN112, Dual LCK/SRC inhibitor) is a potent and orally active Lck/Src inhibitor with IC50s of 2 nM and 6 nM in cell-free assays, respectively. Exhibits >300-fold selectivity against p38α and KDR. Also potently inhibits SIK (IC50 values are 10, 22 and 60 nM for SIK 1, 2 and 3 respectively) and displays selectivity over a range of closely related kinases.
Storage Conditions
2 years -80 in solvent

Related Products

CatalogName
C12131-01Grapiprant (CJ-023,423)
C109004,4'-Dimethoxybenzil
C110204,4'-DDE
C111774,4'-Bis (4-aminophenoxy) biphenyl
C08397-014-Methylumbelliferone (4-MU)
C14473-014-HNE (4-Hydroxynonenal)
C049184,4'-dibromobiphenyl-d8
C167284-Methylumbelliferone (4-MU)
C04114Dimethyl biphenyl-4,4'-dicarboxylate
C09439-014-PBA (4-Phenylbutyric acid)

Alternative Products

CatalogName
MBS576518WH-4-023
MBS386399-01WH 4-023
A14117-2WH 4-023 2mg
A14117-50WH 4-023 50mg
A14117-100WH 4-023 100mg
A14117-5WH 4-023 5mg
A14117-10WH 4-023 10mg

Popular Products