PKI-402

• CAS Number :

  1173204-81-3

• SKU :

  C17035-10mg

• Target :

  PI3K

• Applications :

  PI3K/Akt/mTOR

• Smiles :

  CCN1C2=C (C (=NC (=N2) C3=CC=C (C=C3) NC (=O) NC4=CC=C (C=C4) C (=O) N5CCN (CC5) C) N6CCOCC6) N=N1

• Molecular Formula :

  C29H34N10O3

• Additionnal Information :

  PKI-402 is a potent dual pan-PI3K/mTOR inhibitor targeting PI3Kα/β/γ/δ and mTOR with IC50 of 2 nM/7 nM/16 nM/14 nM and 3 nM, respectively; also potent to PI3Kα mutants E545K and H1047R.

• Storage Conditions :

  2 years -80 in solvent