BMS-536924

CAT: 1568-C16058-01Size: 10 mgDry Ice: YesHazardous: No
CAT#:1568-C16058-01Size:10 mg
Selected
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
CAS Number
468740-43-4
Synonyms
CS-0117
SKU
C16058-10mg
Target
IGF-1R
Applications
Protein Tyrosine Kinase
Smiles
CC1=CC (=CC2=C1N=C (N2) C3=C (C=CNC3=O) NCC (C4=CC (=CC=C4) Cl) O) N5CCOCC5
Molecular Formula
C25H26ClN5O3
Additionnal Information
BMS-536924 (CS-0117) is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for Mek, Fak, and Lck with very little activity for Akt1, MAPK1/2.
Storage Conditions
2 years -80 in solvent

Popular Products