NS 1738
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


NS 1738
CAS Number :
501684-93-1Synonyms :
NSC 213859SKU :
C15979-25mgTarget :
AChRApplications :
Neuronal SignalingSmiles :
C1=CC (=C (C=C1C (F) (F) F) NC (=O) NC2=C (C=CC (=C2) Cl) O) ClMolecular Formula :
C14H9Cl2F3N2O2Additionnal Information :
NS 1738 (NSC 213859) is a novel positive allosteric modulator of the α7 nicotinic acetylcholine receptor (α7 nAChR), with respect to positive modulation of Xenopus laevis oocyte α7 nAChR with EC50 of 3.4 μM, as well as a comparable efficacy at the rat α7 nAChR with EC50 of 3.9 μM.Storage Conditions :
3 years -20°C powder

