INCB054329

CAT: 1568-C13641-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:1568-C13641-01Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1628607-64-6
SKU
C13641-5mg
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1=C (C (=NO1) C) C2=C3C4=C (C=C2) NC (=O) N4C (CO3) C5=CC=CC=N5
Molecular Formula
C19H16N4O3
Additionnal Information
INCB054329 is a structurally distinct bromodomain and extraterminal domain (BET) inhibitor with IC50 values of 44 nM, 5 nM, 9 nM, 1 nM, 28 nM, 3 nM, 119 nM and 63 nM for BRD2-BD1, BRD2-BD2, BRD3-BD1, BRD3-BD2, BRD4-BD1, BRD4-BD2, BRDT-BD1 and BRDT-BD2, respectively.
Storage Conditions
3 years -20°C powder

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