CPI-637

• CAS Number :

  1884712-47-3

• SKU :

  C13252-10mg

• Target :

  Epigenetic Reader Domain

• Applications :

  Epigenetics

• Smiles :

  CC1CC (=O) NC2=CC=CC (=C2N1) C3=CC4=C (C=C3) N (N=C4C5=CN (N=C5) C) C

• Molecular Formula :

  C22H22N6O

• Additionnal Information :

  CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibitor with IC50 values of 0.03 μM and 0.051μM for CBP and EP300 respectively in TR-FRET assay. It is highly selective against other bromodomains, displaying substantial biochemical activity only against BRD9.

• Storage Conditions :

  2 years -80 in solvent