PF-3758309
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: Yes


PF-3758309
CAS Number :
898044-15-0Synonyms :
PF-03758309SKU :
C12436-10mgTarget :
PAKApplications :
Cytoskeletal SignalingSmiles :
CC1=NC2=C (C (=N1) NC3=NNC4=C3CN (C4 (C) C) C (=O) NC (CN (C) C) C5=CC=CC=C5) SC=C2Molecular Formula :
C25H30N8OSAdditionnal Information :
PF-03758309 (PF-03758309) is a potent, ATP-competitive, pyrrolopyrazole inhibitor of PAK4 with Kd of 2.7 nM. PF-3758309 is antiproliferative and induces apoptosis in a HCT116 tumor model.Storage Conditions :
2 years -80 in solvent

