CCG215022

CAT: 1568-C12063-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:1568-C12063-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1813527-81-9
SKU
C12063-1mg
Target
GRK
Applications
GPCR & G Protein
Smiles
CC1=C (C (NC (=O) N1) C2=CC (=C (C=C2) F) C (=O) NCC3=CC=CC=N3) C (=O) NC4=CC5=C (C=C4) NN=C5
Molecular Formula
C26H22FN7O3
Additionnal Information
CCG215022 serves as a pan-G protein-coupled receptor kinases (GRKs) inhibitor with IC50 of 3.9 μM, 0.15 μM, 0.38 μM for GRK1, GRK2, GRK5, respectively.
Storage Conditions
3 years -20°C powder

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