BMS-986020

• CAS Number :

  1257213-50-5

• Synonyms :

  AM152, AP-3152 free acid

• SKU :

  C09424-5mg

• Target :

  LPA Receptor

• Applications :

  GPCR & G Protein

• Smiles :

  CC (OC (=O) NC1=C (ON=C1C) C2=CC=C (C=C2) C3=CC=C (C=C3) C4 (CC4) C (O) =O) C5=CC=CC=C5

• Molecular Formula :

  C29H26N2O5

• Additionnal Information :

  BMS-986020 (AM152, AP-3152 free acid) is a potent and selective antagonist of lysophosphatidic acid receptor 1 (LPA1) . BMS-986020 inhibits bile acid and phospholipid transporters with IC50 of 4.8 μM, 6.2 μM, and 7.5 μM for BSEP, MRP4, and MDR3, respectively. BMS-986020 has the potential for the treatment of idiopathic pulmonary fibrosis (IPF) .

• Storage Conditions :

  3 years -20°C powder