Products for Research Use Only

VU0238429

CAT: 1568-C08749-01Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:1568-C08749-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
1160247-92-6
Synonyms
M5 PAM
SKU
C08749-5mg
Target
AChR
Applications
Neuronal Signaling
Smiles
COC1=CC=C (C=C1) CN2C3=C (C=C (C=C3) OC (F) (F) F) C (=O) C2=O
Molecular Formula
C17H12F3NO4
Additionnal Information
VU0238429 (M5 PAM) is the first positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5/M5) with EC50 of 1.16 μM at M5 and both > 30 μM at M1 and M3. VU0238429 shows no potentiator activity at M2 or M4.
Storage Conditions
3 years -20°C powder

Alternative Products