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Ninerafaxstat trihydrochloride

CAT: 1568-C01891-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:1568-C01891-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2311824-72-1
Synonyms
MB-1018972 trihydrochloride, IMB-101 trihydrochloride
SKU
C01891-5mg
Target
Mitochondrial Metabolism
Applications
Metabolism
Additionnal Information
Ninerafaxstat trihydrochloride (MB-1018972 trihydrochloride, IMB-101 trihydrochloride) acts as a competitive inhibitor of 3-ketoacyl-CoA thiolase (3-KAT) to partially suppress fatty acid oxidation. It is an orally active cardiac mitochondrial drug that restores myocardial energy homeostasis. Ninerafaxstat trihydrochloride regulates myocardial substrate utilization and improves cardiac efficiency. Ninerafaxstat trihydrochloride is also used in research of cardiovascular diseases.

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