Hydroxy Varenicline

• UNSPSC Description:

  Hydroxy varenicline (2-Hydroxyvarenicline) is a metabolite of varenicline (HY-10019), a nicotinic acetylcholine receptor (nAChR) agonist.

• Target Antigen:

  nAChR

• Type:

  Reference compound

• Related Pathways:

  Membrane Transporter/Ion Channel;Neuronal Signaling

• Field of Research:

  Neurological Disease

• Assay Protocol:

  https://www.medchemexpress.com/hydroxy-varenicline.html

• Smiles:

  O=C1NC(C=C(C2=C3)C4CNCC2C4)=C3N=C1

• Molecular Weight:

  227.26

• References & Citations:

  [1]Obach, et al. Metabolism and disposition of varenicline, a selective α4β2 acetylcholine receptor partial agonist, in vivo and in vitro. Drug. Metab. Dispos. 34(1), 121-130 (2006).

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  357424-21-6