Products for Research Use Only

Pexacerfont (Standard)

CAT: 0804-HY-12127RSize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-12127RSize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Pexacerfont (Standard) is the analytical standard of Pexacerfont. This product is intended for research and analytical applications. Pexacerfont is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1±0.6 nM for human CRF1 receptor.
CAS Number
459856-18-9
UNSPSC
12352100
Target
CRFR; Reference Standards
Related Pathways
GPCR/G Protein; Others
Field of Research
Neurological Disease; Endocrinology
Smiles
CC[C@H](NC1=NC(C)=NC2=C(C3=CC=C(OC)N=C3C)C(C)=NN21)C
Molecular Formula
C18H24N6O
Molecular Weight
340.42
References & Citations
[1]Zhou L, et al. In vitro and in vivo metabolism and pharmacokinetics of BMS-562086, a potent and orally bioavailable corticotropin-releasing factor-1 receptor antagonist. Drug Metab Dispos. 2012 Jun;40 (6) :1093-103.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards