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GSK6853 (Standard)

CAT: 0804-HY-100220RSize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-100220RSize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GSK6853 (Standard) is the analytical standard of GSK6853. This product is intended for research and analytical applications. GSK6853, a chemical probe, is a potent and selective inhibitor of the BRPF1 bromodomain. GSK6853 shows excellent BRPF1 potency (pKd = 9.5) and greater than 1600-fold selectivity over all other bromodomains[1].
CAS Number
1910124-24-1
Target
Epigenetic Reader Domain; Reference Standards
Related Pathways
Epigenetics; Others
Field of Research
Cancer
Smiles
C[C@@H]1CNCCN1C2=C(NC(C3=CC=CC=C3OC)=O)C=C(C(N4C)=C2)N(C)C4=O
Molecular Formula
C22H27N5O3
Molecular Weight
409.48
References & Citations
[1]Bamborough P et al. GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain. ACS Med Chem Lett. 2016 May 9;7 (6) :552-7.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards

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Alternative Products

CatalogName
BUP13485-01GSK6853
A16330-50GSK6853 50mg
A16330-2GSK6853 2mg
A16330-200GSK6853 200mg
A16330-10GSK6853 10mg
A16330-5GSK6853 5mg
A16330-100GSK6853 100mg
A16330-25GSK6853 25mg
TBI4016-25MGGSK6853, BRPF1 inhibitor
A16330-10mM-DGSK6853 10mM * 1mL in DMSO

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