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CREBBP-IN-1

CAT: 0804-HY-114971Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-114971Size:1 Each
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CREBBP-IN-1 (Compound 10) exhibits good affinity with CREBBP bromodomain with Kd of 0.77 μM[1].
CAS Number
[1801324-41-3]
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/crebbp-in-1.html
Smiles
O=C(C1=CC=CC(C(NC2=CC(C(C)=O)=CC=C2OCC)=O)=C1)O
Molecular Formula
C18H17NO5
Molecular Weight
327.33
References & Citations
[1]Xu M, et al., Discovery of CREBBP Bromodomain Inhibitors by High-Throughput Docking and Hit Optimization Guided by Molecular Dynamics. J Med Chem. 2016 Feb 25;59 (4) :1340-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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