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CMPD101 hydrochloride

CAT: 0931-T89364-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T89364-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1941168-71-3
Bioactivity
CMPD101 hydrochloride is a membrane-permeable small molecule inhibitor of GRK2 and GRK3, exhibiting IC50 values of 18 nM and 5.4 nM, respectively. This compound also inhibits Rho-associated kinase 2 (ROCK-2) and PKCα, with IC50 values of 1.4 μM and 8.1 μM, respectively.
Smiles
Cl.O=C(NCC=1C=CC=CC1C(F)(F)F)C=2C=CC=C(C2)NCC3=NN=C(C=4C=CN=CC4)N3C
Molecular Formula
C24H22ClF3N6O
Molecular Weight
502.92
Shipping Conditions
Ice Packs
Storage Temperature
-20°C