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VD4162

CAT: 0931-T87610-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T87610-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2574390-19-3
Target
Serine Protease
Related Pathways
Proteases/Proteasome
Bioactivity
VD4162 (Compound 8b), a macrocyclic inhibitor of serine proteases, exhibits enhanced potency against four key target enzymes: TMPRSS2 (IC 50 = 3.7 nM), HGFA (IC 50 = 3.3 nM), matriptase (IC 50 = 2.9 nM), and hepsin (IC 50 = 0.54 nM) . This compound is utilized in cancer research [1].
Smiles
C(C=1C=2C(NC1)=CC=CC2)[C@H]3NC(=O)[C@@H](NC(C)=O)CC=4C=CC(=CC4)OCCCC[C@@H](C(N[C@H](C(=O)C5=NC=6C(S5)=CC=CC6)CCCNC(=N)N)=O)NC3=O
Molecular Formula
C41H47N9O6S
Molecular Weight
793.93
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
HY-161370VD4162