Rezatapopt

• Target :

  Others|||MDM-2/p53|||p53

• Related Pathways :

  Others|||Apoptosis

• Purity :

  0.9812

• Bioactivity :

  Rezatapopt (PC14586) is a small molecule p53 reactivator with anti-tumor activity that selectively binds to the cleft present in the TP53 Y220C mutant protein and restores the p53 wild-type (normal) conformation and transcriptional activity, and can be used to study locally advanced or metastatic solid tumors.

• Smiles :

  N(C1=C2C(N(CC(F)(F)F)C(C#CCNC3=C(OC)C=C(C(NC)=O)C=C3)=C2)=CC=C1)[C@H]4[C@@H](F)CN(C)CC4

• Molecular Formula :

  C28H31F4N5O2

• Molecular Weight :

  545.57

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2636846-41-6