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Rezatapopt

CAT: 0931-T81289-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T81289-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2636846-41-6
Target
Others, MDM-2/p53, p53
Related Pathways
Others, Apoptosis
Purity
0.9812
Bioactivity
Rezatapopt (PC14586) is a small molecule p53 reactivator with anti-tumor activity that selectively binds to the cleft present in the TP53 Y220C mutant protein and restores the p53 wild-type (normal) conformation and transcriptional activity, and can be used to study locally advanced or metastatic solid tumors.
Smiles
N(C1=C2C(N(CC(F)(F)F)C(C#CCNC3=C(OC)C=C(C(NC)=O)C=C3)=C2)=CC=C1)[C@H]4[C@@H](F)CN(C)CC4
Molecular Formula
C28H31F4N5O2
Molecular Weight
545.57
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
M37295-01Rezatapopt

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