WAY-649123

CAT: 0931-T80787-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0931-T80787-01Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
801244-46-2
Target
Others
Related Pathways
Others
Bioactivity
WAY-649123 is an active molecule that exhibits (in vitro) antagonistic properties against (alpha-1A adrenergic receptors), with a (pKi) of 8.9. It also demonstrates a 70-fold selectivity over (alpha-1B) and 100-fold selectivity over (alpha-1D) subtypes. This compound has been shown to cross the blood-brain barrier (BBB) effectively in preclinical trials. Furthermore, WAY-649123 exhibits a high level of oral bioavailability and a favorable pharmacokinetic profile, making it a potential candidate for clinical development targeting conditions associated with (alpha-1A) receptors.
Smiles
O=C(NC1=CC=C(F)C=C1F)CC2=CC=C3OCCOC3=C2
Molecular Formula
C16H13F2NO3
Molecular Weight
305.28
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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