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Targefrin

CAT: 0931-T76375-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T76375-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Ephrin Receptor
Related Pathways
Tyrosine Kinase/Adaptors
Bioactivity
Targefrin is a potent antagonist targeting EphA2, exhibiting a dissociation constant of 21 nM and an IC50 value of 10.8 nM for the EphA2-LBD. It promotes receptor internalization and degradation across multiple pancreatic cancer cell lines [1].
Molecular Formula
C85H116F3N19O15
Molecular Weight
1700.94
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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