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Desmethylazelastine

CAT: 0931-T74583-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T74583-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
47491-38-3
Target
Others, Drug Metabolite
Related Pathways
Others, Metabolism
Bioactivity
Desmethylazelastine, the primary active metabolite of Azelastine, undergoes oxidative metabolism via the cytochrome P450 enzyme system, exhibits a 97% protein binding rate, and has an elimination half-life of 54 hours. Azelastine, an orally active, selective, and high-affinity histamine H1-receptor antagonist, is utilized in the research of allergic rhinitis, asthma, diabetic hyperlipidemia, and SARS-CoV-2 [1] [2] [3] [4] [5].
Smiles
Clc1ccc(Cc2nn(C3CCCNCC3)c(=O)c3ccccc23)cc1
Molecular Formula
C21H22ClN3O
Molecular Weight
367.87
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
HY-147336-01Desmethylazelastine

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