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YM458

CAT: 0931-T74542-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T74542-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2770108-93-3
Target
Histone Methyltransferase, Apoptosis, Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic, Apoptosis
Bioactivity
YM458, a potent dual inhibitor of EZH2 and BRD4, exhibits IC50 values of 490 nM and 34 nM, respectively. This compound effectively hinders cell proliferation and colony formation, while also inducing cell cycle arrest and apoptosis in solid tumor cells, making it a viable candidate for anticancer research [1].
Molecular Formula
C53H61ClN8O5S
Molecular Weight
957.62
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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