Products for Research Use Only

EGFR-IN-42

CAT: 0931-T74457-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T74457-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Target
Others, EGFR
Related Pathways
JAK/STAT signaling, Angiogenesis, Others, Tyrosine Kinase/Adaptors
Bioactivity
EGFR-IN-42 (Compound 17b), a potent EGFR inhibitor, demonstrates single-digit nanomolar activity by covalently linking tamoxifen or endoxifen with gefitinib, retaining both ER antagonist activity and EGFR inhibition, resulting in superior anti-cancer activity [1].
Molecular Formula
C49H53ClFN5O5
Molecular Weight
846.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C