TrkA-IN-3
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


TrkA-IN-3
Target:
Others|||Trk receptorRelated Pathways:
Tyrosine Kinase/Adaptors|||OthersBioactivity:
TrkA-IN-3 is a potent, subselective, and allosteric inhibitor of TrkA with an IC50 of 22.4 nM, demonstrating over 8000-fold selectivity towards TrkA compared to TrkB and TrkC, making it valuable for pain research.Smiles:
CN1C=CC(=N1)C2=C(C=CC(=C2)C(=O)NC3=C(N=CC(=C3)C(=O)O)C4=CC=CC=C4)C(F)(F)FMolecular Formula:
C24H17F3N4O3Molecular Weight:
466.41Shipping Conditions:
Cool packStorage Temperature:
-20°C
