(R) -HH2853

• Target:

  Histone Methyltransferase

• Related Pathways:

  Chromatin/Epigenetic

• Purity:

  >99.99%

• Bioactivity:

  (R) -HH2853 is a potent EZH2 inhibitor with an IC50 <100 nM for EZH2-Y641F. (R) -HH2853 has anticancer and antitumor activity and can be used in autoimmune diseases.

• Smiles:

  [C@@H](C)(C=1N2C(=C(C=C2)C3=CC=C(C)N=N3)C=C(C(NCC4=C(OC)C=C(C)NC4=O)=O)C1C)N5CCN(CC(F)(F)F)CC5

• Molecular Formula:

  C31H36F3N7O3

• Molecular Weight:

  611.66

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2202678-06-4