Products for Research Use Only

PF-04479745 tartrate

CAT: 0931-T70379-01Size: 25 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T70379-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
1613691-76-1
Target
Others
Related Pathways
Others
Bioactivity
PF-04479745, also known as PF-4479745, is a potent and selective 5-HT2C agonist (EC50 = 10 nM) . PF-4479745 displayed robust pharmacology in a preclinical canine model of stress urinary incontinence (SUI) and no measurable functional agonism at the key selectivity targets 5-HT2A and 5-HT2B in relevant tissue-based assay systems.
Smiles
O[C@H]([C@@H](O)C(O)=O)C(O)=O.CNc1nc(Cc2ccccc2)nc2[C@@H](C)CNCCc12
Molecular Formula
C21H28N4O6
Molecular Weight
432.477
Shipping Conditions
Ice Packs
Storage Temperature
-20°C