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SKF89976A HCl

CAT: 0931-T68550-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T68550-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
85375-85-5
Target
GABA Receptor, Others
Related Pathways
Neuroscience, Others, Membrane transporter/Ion channel
Bioactivity
SKF89976A is a potent GABA uptake inhibitor, which is selective for GAT-1 (IC50 values are 0.13, 550, 944 and 7210 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively) . SKF89976A inhibits transport current competitively (Ki = 7 μM) and transmitter-gated current non-competitively (Ki = 0.03 nM) . It is able to pass the blood-brain barrier after systemic administration and is active in vivo.
Smiles
C(=CCCN1CC(C(O)=O)CCC1)(C2=CC=CC=C2)C3=CC=CC=C3
Molecular Formula
C22H25NO2
Molecular Weight
335.44
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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HY-100228A-01SKF89976A (hydrochloride)
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