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UPSEM792

CAT: 0931-T209079-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T209079-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2323525-19-3
Target
5-HT Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Bioactivity
UPSEM792 is a pharmacologically selective agonist molecule (PSEM) for PSAM4-GlyR, with an affinity Ki of 0.7 nM. It acts as a substrate for efflux transporters in both wild-type mice brains and in P-gp and BCRP double knockout mice. Additionally, uPSEM792 may serve as a lead compound in the development of PET radioligands for PSAM4-GlyR.
Smiles
O=C1C=NC=2C=C3C(=CC2N1C)C4CNCC3C4
Molecular Formula
C14H15N3O
Molecular Weight
241.29
Shipping Conditions
Ice Packs
Storage Temperature
-20°C