Products for Research Use Only

Blixeprodil

CAT: 0931-T206599-01Size: 10 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T206599-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
2881017-49-6
Target
IGluR
Related Pathways
Neuroscience, Membrane transporter/Ion channel
Bioactivity
Blixeprodil (GM-1020) is an orally active NMDA receptor antagonist with an affinity of Ki = 3.25 μM in rat cortical tissue. It inhibits NR1/2A-NMDAR-mediated currents in HEK293 cells with an IC50 of 1.192 μM. Blixeprodil demonstrates antidepressant effects in rat models and exhibits blood-brain barrier permeability.
Smiles
N(C)[C@@]1(C(=O)CCCC1)C2=CC=C(F)C=C2
Molecular Formula
C13H16FNO
Molecular Weight
221.271
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products