Products for Research Use Only

Darlifarnib

CAT: 0931-T206317-01Size: 10 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T206317-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
2939824-30-1
Target
Transferase
Related Pathways
Metabolism
Bioactivity
Darlifarnib (Compound (S) -058) is an inhibitor of farnesyl transferase and geranylgeranyltransferase, with IC50 values of ≤ 10 nM and > 1000 nM, respectively. It exhibits high metabolic stability in human and mouse liver microsomes, with a half-life of over 100 minutes.
Smiles
N#CC=1N=C2C=CC3=CC2=C(C1)C=4C=CC=C(OCC5=CC(=CC=C5C#N)C3(N)C6=CN=CN6C)C4
Molecular Formula
C29H20N6O
Molecular Weight
468.509
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products