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A-800141

CAT: 0931-T204983-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T204983-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
681245-85-2
Target
Aminopeptidase
Related Pathways
Metabolism
Bioactivity
A-800141 is an orally active and selective MetAP2 inhibitor with an IC50 of 12 nM, while showing weaker inhibitory activity against MetAP1 (IC50: 36 μM) . GAPDH can serve as a biomarker for monitoring the inhibition of MetAP2 by A-800141. This compound exhibits anti-angiogenic and anticancer properties in various xenograft tumor models.
Smiles
C(O)(=O)C1=C2C(=CC=C1NS(=O)(=O)C3=C(/C=C\CN(CC)CC)C=CC=C3)CCCC2
Molecular Formula
C24H30N2O4S
Molecular Weight
442.571
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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CatalogName
HY-119062A-800141

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