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Cetagliptin

CAT: 0931-T203104-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T203104-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2243737-33-7
Target
Cytochromes P450, Proteasome, P-gp
Related Pathways
Membrane transporter/Ion channel, Ubiquitination, Metabolism, Neuroscience, Proteases/Proteasome
Bioactivity
Cetagliptin is an orally active inhibitor of dipeptidyl peptidase 4 (DPP-4) and CYP2D6, with an IC50 of 6 μM. It acts as a substrate for P-glycoprotein and helps reduce GLP-1 degradation, maintaining postprandial blood glucose levels. It is used in research for type 2 diabetes.
Smiles
P(=O)(O)(O)O.C(F)(F)(F)C=1N2C([C@@H](C)N(C(C[C@@H](CC3=C(F)C=C(F)C(F)=C3)N)=O)CC2)=CN1
Molecular Formula
C18H21F6N4O5P
Molecular Weight
518.35
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
HY-170569Cetagliptin

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