RR-49

• Bioactivity :

  RR-49 is an innovative difluorinated analogue. This compound demonstrates exceptional pH sensitivity, showing the same efficacy for DAMGO in MOR cAMP assays at pH 6.5 as it does at pH 7.4, but with a 19-fold increase in potency (IC50) . It holds significant promise as an analgesic for treating inflammatory pain with a lower potential for abuse.

• Smiles :

  O=C(N(C=1C=CC=CC1)C2CCN(CC2)CC(F)C=3C=CC=CC3F)CC

• Molecular Formula :

  C22H26F2N2O

• Molecular Weight :

  372.45

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2376328-79-7