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Enrasentan edamine

CAT: 0931-T201997-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T201997-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
183507-63-3
Bioactivity
Enrasentan (also known as SB-217242) is a dual receptor endothelin antagonist with a higher affinity for the ET (A) receptor. In animal models of hypertension and cardiac hypertrophy, this compound reduces blood pressure, prevents cardiac hypertrophy, and preserves myocardial function. Enrasentan enhances survival rates, limits left ventricular remodeling, and maintains myocardial performance in hypertensive cardiac hypertrophy and dysfunction.
Smiles
NCCN.OC([C@H]1[C@H](C2=C(C=C(C=C2)OC)OCCO)C3=CC(OCCC)=CC=C3[C@@H]1C4=CC=C(OCO5)C5=C4)=O.OC([C@H]6[C@H](C7=C(C=C(C=C7)OC)OCCO)C8=CC(OCCC)=CC=C8[C@@H]6C9=CC=C(OCO%10)C%10=C9)=O
Molecular Formula
C30H34NO8
Molecular Weight
536.6
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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