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XE991 dihydrochloride

CAT: 0957-S2967Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0957-S2967Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
XE 991 (LS190926) dihydrochloride is a blocker of Kv7 (KCNQ) channels that potently inhibits KCNQ1 (Kv7.1), KCNQ2 (Kv7.2), KCNQ2 + KCNQ3 (Kv7.3) channel, and M-current with IC50 of 0.75 μM, 0.71 μM, 0.6 μM, and 0.98 μM, respectively.
CAS Number
122955-13-9
Synonyms
LS190926 dihydrochloride
Target
Potassium Channel
Activity
Transmembrane Transporters
Molecular Formula
C26H22Cl2N2O
Storage Conditions
3 years -20°C powder