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Gefitinib-based PROTAC 3

CAT: 0957-S0070-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-S0070-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Gefitinib-based PROTAC 3 which conjugates an EGFR binding element to a VHL ligand via a linker induces degradation of EGFR and mutants with DC50 of 11.7 nM and 22.3 nM in HCC827 (Exon 19 del) and H3255 (L858R) cells, respectively.
CAS Number
2230821-27-7
Target
EGFR
Activity
Protein Tyrosine Kinase
Molecular Formula
C47H57ClFN7O8S
Storage Conditions
3 years -20°C powder

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